SCHEMBL3658121

SCHEMBL3658121

COC(=O)CCC(=O)c1c(CC(=O)COc2ccc(Oc3ccc(C(F)(F)F)cc3)cc2)[nH]c2ccc(C(=O)OC)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KIF11 P52732 1/20 0.38
BCHE P06276 1/20 0.36
GRM4 Q14833 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
AKR1C3 P42330 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
TRPV1 Q8NER1 1/20 0.35
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPT P10636 3/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658319 0.85 MEN1 (0.43) MEN1KMT2ALMNAATML3MBTL1
SCHEMBL3653066 0.80 KMT2A (0.48) MEN1KMT2ALMNAATML3MBTL1
SCHEMBL3658581 0.77 PLA2G4A (0.46) MEN1KMT2AATML3MBTL1MDH1
SCHEMBL3657841 0.69 PLA2G4A (0.50) MEN1KMT2AATML3MBTL1MDH1
SCHEMBL2807365 0.69 PLA2G4A (0.59)
SCHEMBL3656549 0.68 PLA2G4A (0.44)
SCHEMBL23606009 0.68 ALDH1A1 (0.59) LMNAGRM4ALDH1A1PPARGPPARD
SCHEMBL13127472 0.67 PLA2G4A (0.46) AKR1C3
SCHEMBL1782842 0.67 LMNA (0.69) MEN1KMT2ALMNATRPV1KDM4E
SCHEMBL2806998 0.66 AKR1C3 (0.39) KMT2ALMNAAKR1C3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215059-A2 NOVEL HETEROARYL-SUBSTITUTED ACETONE DERIVATIVE, SUITABLE FOR INHIBITING PHOSPHOLIPASE A2 Westfälische Wilhelms-Universität Münster (DE) 2010-08-11 EP disclosed
WO-2009040314-A2 NOVEL HETEROARYL-SUBSTITUTED ACETONE DERIVATIVES, SUITABLE FOR INHIBITING PHOSPHOLIPASE A2 Westfälische Wilhelms Universität Münster (DE) 2009-04-02 WO disclosed