SCHEMBL3658163

SCHEMBL3658163

CC(C)(C)c1ccc(S(=O)(=O)Nc2ccsc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.59
UQCRB P14927 3/20 0.59
MEN1 O00255 2/20 0.59
MAPT P10636 2/20 0.59
KMT2A Q03164 2/20 0.59
CA1 P00915 2/20 0.59
CA2 P00918 2/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C19 P33261 1/20 0.59
HDAC3 O15379 2/20 0.54
HDAC11 Q96DB2 2/20 0.54
HDAC8 Q9BY41 2/20 0.54
HDAC6 Q9UBN7 2/20 0.54
POLB P06746 2/20 0.54
HTT P42858 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
RORA P35398 1/20 0.54
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL812679 0.81 ALDH1A1 (0.83) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL3934185 0.78 KEAP1 (0.62) ALDH1A1MEN1MAPTKMT2ACA1
SCHEMBL12042475 0.77 ALDH1A1 (0.71) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL13433558 0.76 ALDH1A1 (0.73) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL30014158 0.76 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL1040954 0.76 ALDH1A1 (0.73) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL7178237 0.74 UQCRB (1.00) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL20657557 0.74 KMT2A (1.00) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL12042479 0.74 ALDH1A1 (0.76) ALDH1A1UQCRBMEN1MAPTKMT2A
SCHEMBL95623 0.74 ALDH1A1 (0.71) ALDH1A1UQCRBMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220065-A2 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-08-25 EP disclosed
WO-2009017719-A2 MODULATORS OF CCR9 RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-02-05 WO disclosed