SCHEMBL365894

SCHEMBL365894

CCCCOC(=O)c1c2ccccc2n2cc(O)ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.48
MAPK1 P28482 3/20 0.48
LMNA P02545 3/20 0.48
ESR1 P03372 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
NR1H2 P55055 1/20 0.48
RNASEL Q05823 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
EGFR P00533 1/20 0.46
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 7/20 0.43
CYP3A4 P08684 2/20 0.43
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366765 0.96 TSHR (0.48) TSHRMAPK1LMNAESR1CYP1A2
SCHEMBL365400 0.93 ELANE (0.47) TSHRLMNAESR1SMN1; SMN2TDP1
SCHEMBL364761 0.87 KDM4E (0.52) TSHRMAPK1LMNACYP1A2SMN1; SMN2
SCHEMBL366754 0.86 TSHR (0.45) TSHRMAPK1LMNAESR1CYP1A2
SCHEMBL366408 0.84 ALDH1A1 (0.52) L3MBTL1TDP1EGFRKDM4EALDH1A1
SCHEMBL367540 0.81 PSEN1 (0.45) TSHRMAPK1LMNACYP1A2CYP2C19
SCHEMBL366763 0.81 ALDH1A1 (0.44) TSHRMAPK1LMNACYP1A2L3MBTL1
SCHEMBL365893 0.81 ALDH1A1 (0.53) TSHRMAPK1LMNAESR1CYP1A2
SCHEMBL364931 0.80 NR4A2 (0.50) LMNACYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL366392 0.80 PSEN1 (0.46) TSHRMAPK1LMNAL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed