SCHEMBL366765

SCHEMBL366765

CCCCCOC(=O)c1c2ccccc2n2cc(O)ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.48
MAPK1 P28482 3/20 0.48
TP53 P04637 1/20 0.48
CYP3A4 P08684 1/20 0.48
ALDH1A1 P00352 6/20 0.47
LMNA P02545 4/20 0.47
KDM4E B2RXH2 5/20 0.45
HSD17B10 Q99714 2/20 0.45
HPGD P15428 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
HTT P42858 1/20 0.44
ESR1 P03372 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
NR1H2 P55055 1/20 0.44
RNASEL Q05823 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4A O75164 1/20 0.43
KDM4C Q9H3R0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365894 0.96 TSHR (0.48) TSHRMAPK1TP53CYP3A4ALDH1A1
SCHEMBL365400 0.91 ELANE (0.47) TSHRALDH1A1LMNAKDM4EHPGD
SCHEMBL364761 0.86 KDM4E (0.52) TSHRMAPK1CYP3A4ALDH1A1LMNA
SCHEMBL366408 0.83 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDL3MBTL1TDP1
SCHEMBL366754 0.82 TSHR (0.45) TSHRMAPK1TP53CYP3A4ALDH1A1
SCHEMBL366764 0.81 ALDH1A1 (0.50) TSHRMAPK1TP53CYP3A4ALDH1A1
SCHEMBL366392 0.81 PSEN1 (0.46) TSHRMAPK1TP53CYP3A4ALDH1A1
SCHEMBL364931 0.79 NR4A2 (0.50) CYP3A4ALDH1A1LMNAKDM4EHSD17B10
SCHEMBL367016 0.79 TSHR (0.42) TSHRMAPK1TP53CYP3A4ALDH1A1
SCHEMBL365562 0.78 CYP3A4 (0.46) TSHRTP53CYP3A4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed