SCHEMBL3660176

SCHEMBL3660176

O=C1Cc2cc(C(=O)Nc3ccccc3)ccc2N1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 14/20 0.58
HDAC3 O15379 1/20 0.58
PTPN1 P18031 2/20 0.51
TRPV1 Q8NER1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31139504 1.00 SMYD3 (0.58) SMYD3HDAC3PTPN1TRPV1
SCHEMBL23143565 0.89 TRPV1 (0.56) SMYD3HDAC3PTPN1TRPV1
SCHEMBL5842454 0.86 TLK2 (0.57) SMYD3HDAC3PTPN1
SCHEMBL4415749 0.82 TLK2 (0.56) SMYD3HDAC3
SCHEMBL396708 0.82 KCNK3 (0.57) SMYD3TRPV1
SCHEMBL3193164 0.80 SMYD3 (0.61) SMYD3
SCHEMBL26547572 0.80 SMYD3 (0.56) SMYD3HDAC3
SCHEMBL3195105 0.80 CRBN (0.68) SMYD3HDAC3
SCHEMBL19691220 0.80 SMYD3 (0.61) SMYD3HDAC3
SCHEMBL16048824 0.80 SMYD3 (0.67) SMYD3HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12528797-B2 Heterocyclic compounds for medical treatment C4 THERAPEUTICS, INC. 2026-01-20 US disclosed
EP-4470618-A2 HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT C4 Therapeutics, Inc. (US) 2024-12-04 EP disclosed
EP-3935050-B1 HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT C4 THERAPEUTICS INC (US) 2024-10-02 EP disclosed
US-11787802-B2 Dihydrobenzimidazolones for medical treatment C4 THERAPEUTICS, INC. (US) 2023-10-17 US disclosed
US-20230019060-A1 HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT C4 THERAPEUTICS, INC. (US) 2023-01-19 US disclosed
US-20230019060-A1 HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT C4 THERAPEUTICS, INC. (US) 2023-01-19 US disclosed
CN-113557235-A Heterocyclic compounds for use in medical therapy C4医药公司 2021-10-26 CN disclosed
US-8765748-B2 Indazolyl, benzimidazolyl, benzotriazolyl substituted indolinone derivatives as kinase inhibitors useful in the treatment of cancer UNIVERSITY HEALTH NETWORK (CA) 2014-07-01 US disclosed
US-20110065702-A1 INDAZOLYL, BENZIMIDAZOLYL, BENZOTRIAZOLYL SUBSTITUTED INDOLINONE DERIVATIVES AS KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER UNIVERSITY HEALTH NETWORK 2011-03-17 US disclosed
EP-2235004-A1 INDAZOLYL, BENZIMIDAZOLYL, BENZOTRIAZOLYL SUBSTITUTED INDOLMONE DERIVATIVES AS KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER University Health Network (CA) 2010-10-06 EP disclosed
WO-2009079767-A9 INDAZOLYL, BENZIMIDAZOLYL, BENZOTRIAZOLYL SUBSTITUTED INDOLINONE DERIVATIVES AS KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER UNIVERSITY HEALTH NETWORK (CA) 2009-10-01 WO disclosed
WO-2009079767-A1 INDAZOLYL, BENZIMIDAZOLYL, BENZOTRIAZOLYL SUBSTITUTED INDOLINONE DERIVATIVES AS KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER UNIVERSITY HEALTH NETWORK (CA) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230019060-A1 HETEROCYCLIC COMPOUNDS FOR MEDICAL TREATMENT CRBN, MDM2, RBX1 SMYD3 2455/4885HDAC3 1104/4885PTPN1 3411/4885
US-12528797-B2 Heterocyclic compounds for medical treatment CRBN, CUL2, ADRM1 SMYD3 2889/4885HDAC3 537/4885PTPN1 1572/4885
US-20110065702-A1 INDAZOLYL, BENZIMIDAZOLYL, BENZOTRIAZOLYL SUBSTITUTED INDOLINONE DERIVATIVES AS KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER TNNI3K, ABL1, TK1 SMYD3 2681/4885HDAC3 875/4885PTPN1 1506/4885
US-11787802-B2 Dihydrobenzimidazolones for medical treatment CRBN, CUL4A, ADRM1 SMYD3 2716/4885HDAC3 967/4885PTPN1 2783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.