SCHEMBL3661150

SCHEMBL3661150

CC(C)COC(=O)N1CCC(C)(NCc2ccc(C(F)(F)F)nc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.44
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
NAMPT P43490 1/20 0.40
GPR119 Q8TDV5 2/20 0.40
RORC P51449 1/20 0.40
ENPP2 Q13822 9/20 0.39
SCN9A Q15858 2/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNQ4 P56696 1/20 0.38
KCNQ5 Q9NR82 1/20 0.38
ADORA2A P29274 1/20 0.38
SCN5A Q14524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3661148 0.85 GPR119 (0.44) MGLLNAMPTGPR119
SCHEMBL3658892 0.77 HRH3 (0.46) TSHRENPP2
SCHEMBL3714260 0.72 KDM1A (0.43) CYP3A4CYP2C9CYP2C19NAMPT
SCHEMBL14155585 0.70 NAMPT (0.46) MGLLNAMPTENPP2
SCHEMBL3490742 0.69 NAMPT (0.45) MGLLNAMPTENPP2
SCHEMBL15544614 0.68 CYP2D6 (0.39) CYP1A2CYP2D6CYP2C9GPR119RORC
SCHEMBL3494553 0.68 NAMPT (0.44) MGLLNAMPTENPP2
SCHEMBL26081084 0.68 MGLL (0.46) MGLLGPR119
SCHEMBL17269796 0.67 GPR119 (0.54) GPR119
SCHEMBL20778366 0.67 ABHD6 (0.48) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238135-A1 NAPHTHYRIDIN-2(1H) -ONE COMPOUNDS USEFUL AS ANTIBACTERIALS Glaxo Group Limited (GB) 2010-10-13 EP disclosed
WO-2009090222-A1 NAPHTHYRIDIN-2(1H) -ONE COMPOUNDS USEFUL AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2009-07-23 WO disclosed