SCHEMBL3663254

SCHEMBL3663254

COc1ccc2c(O)cc(-c3ccn(C)n3)nc2c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
LRRK2 Q5S007 1/20 0.36
JMJD6 Q6NYC1 4/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
GPR35 Q9HC97 1/20 0.33
RAC1 P63000 2/20 0.32
KDM5B Q9UGL1 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
DNMT1 P26358 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PDE10A Q9Y233 1/20 0.32
AURKA O14965 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3659800 0.80 MEN1 (0.34) KDM4EMEN1KMT2APOLBGAA
SCHEMBL13929789 0.79 PLAU (0.45) LRRK2MAPT
SCHEMBL996497 0.78 CCR1 (0.42) LRRK2MEN1KMT2AGAANPC1
SCHEMBL3657864 0.78 HTR2A (0.37) KDM4EMEN1KMT2APOLBGAA
SCHEMBL3627208 0.77 TDO2 (0.51) KDM4EMEN1KMT2AMAPTSMN1; SMN2
SCHEMBL3625396 0.77 HTT (0.36) KDM4EMEN1KMT2AGAAESR1
SCHEMBL3624833 0.77 ENPP3 (0.43) KDM4EMEN1KMT2APOLBGAA
SCHEMBL15216114 0.76 GAA (0.38) KDM4EMEN1KMT2APOLBGAA
SCHEMBL8083922 0.76 PTGS2 (0.39) KDM4ENPC1MAPTRAB9A
SCHEMBL997481 0.74 ADORA2A (0.33) MEN1KMT2APOLBGAAGPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033466-A1 MACROCYCLIC INHIBITORS OF HEPATITIS C PROTEASE PHENOMIX CORPORATION (US) 2010-03-25 WO disclosed