SCHEMBL3663873

SCHEMBL3663873

N=C(OCCc1ccc2ccccc2c1)C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
PLAU P00749 2/20 0.46
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
SLC13A5 Q86YT5 1/20 0.42
MC4R P32245 1/20 0.42
MC5R P33032 1/20 0.42
PDPK1 O15530 1/20 0.42
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
SOX18 P35713 1/20 0.41
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
PRSS1 P07477 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005477 0.84 CYP1A2 (0.53) CYP1A2PLAUHDAC1HDAC8SLC13A5
SCHEMBL13034170 0.78 CYP1A2 (0.53) CYP1A2HDAC1HDAC8SLC13A5PDPK1
SCHEMBL22920624 0.78 APP (0.49) CYP1A2HDAC1HDAC8SLC13A5PDPK1
Hydrochloric Acid SCHEMBL27558956 0.77 CYP1A2 (0.51) CYP1A2HDAC1HDAC8SLC13A5PDPK1
SCHEMBL3663358 0.77 HTR3E (0.51) CYP3A4
SCHEMBL20809625 0.76 CYP1A2 (0.50) CYP1A2HDAC1HDAC8SLC13A5PDPK1
Hydrochloric Acid SCHEMBL1625284 0.75 PLAU (0.47) CYP1A2PLAUHDAC1HDAC8MC4R
SCHEMBL5267795 0.75 THRB (0.56) CYP1A2HDAC1HDAC8SLC13A5PDPK1
SCHEMBL6934376 0.75 CYP1A2 (0.49) CYP1A2HDAC1HDAC8SLC13A5PDPK1
SCHEMBL3661748 0.74 IDO1 (0.42) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139895-A1 AZA-PYRIDOPYRIMIDINONE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-01-06 EP disclosed
WO-2008116742-A1 AZA-PYRIDOPYRIMIDINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-10-02 WO disclosed