SCHEMBL3661748

SCHEMBL3661748

N=C(OCCc1ccc(F)c(Cl)c1)C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
PIK3CA P42336 1/20 0.40
DAO P14920 1/20 0.38
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RPA1 P27694 1/20 0.36
PNMT P11086 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
YWHAG P61981 1/20 0.35
APP P05067 1/20 0.35
F9 P00740 1/20 0.35
F10 P00742 1/20 0.35
CNR2 P34972 1/20 0.35
GRM2 Q14416 1/20 0.35
GRM3 Q14832 1/20 0.35
ENPP2 Q13822 1/20 0.35
ATXN2 Q99700 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3663358 0.80 HTR3E (0.51) IDO1PNMTTAAR1
Hydrochloric Acid SCHEMBL1623226 0.76 IDO1 (0.37) IDO1PIK3CADAOHDAC3HDAC1
SCHEMBL3662510 0.74 MMP2 (0.39)
SCHEMBL3663873 0.74 CYP1A2 (0.48) HDAC1
SCHEMBL15517814 0.74 PIK3CA (0.47) IDO1PIK3CADAOHDAC3HDAC1
SCHEMBL4847962 0.74 PNMT (0.43) IDO1PIK3CADAOPNMTTAAR1
Hydrochloric Acid SCHEMBL4718123 0.73 PNMT (0.42) IDO1PIK3CADAOPNMTTAAR1
SCHEMBL6917155 0.72 PNMT (0.49) IDO1PNMTTAAR1TSHR
SCHEMBL11716776 0.71 PNMT (0.52) IDO1PNMTTAAR1TSHR
SCHEMBL2791406 0.71 PIK3CA (0.54) IDO1PIK3CAHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139895-A1 AZA-PYRIDOPYRIMIDINONE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-01-06 EP disclosed
WO-2008116742-A1 AZA-PYRIDOPYRIMIDINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-10-02 WO disclosed