SCHEMBL3664535

SCHEMBL3664535

O=C(O)Oc1nc(-c2cccs2)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.56
RAB9A P51151 8/20 0.52
NPC1 O15118 7/20 0.52
MAPT P10636 5/20 0.52
ATM Q13315 2/20 0.52
TP53 P04637 1/20 0.52
SMN1; SMN2 Q16637 4/20 0.50
LMNA P02545 1/20 0.50
FFAR1 O14842 2/20 0.47
HPGD P15428 1/20 0.47
DAGLA Q9Y4D2 1/20 0.47
HDAC1 Q13547 3/20 0.47
HDAC4 P56524 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KDM4E B2RXH2 2/20 0.47
PKM P14618 1/20 0.47
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HDAC2 Q92769 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL492763 0.77 SMN1; SMN2 (0.64) MCL1RAB9ANPC1MAPTATM
SCHEMBL4083201 0.76 NR1H4 (0.52) RAB9ANPC1MAPTTP53SMN1; SMN2
SCHEMBL2162193 0.73 NPC1 (0.70) MCL1RAB9ANPC1MAPTATM
SCHEMBL29518033 0.73 NPC1 (0.61) MCL1RAB9ANPC1MAPTATM
SCHEMBL3666186 0.73 ALDH1A1 (0.43) RAB9ANPC1MAPTLMNAALDH1A1
SCHEMBL6325635 0.71 MCL1 (1.00) MCL1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL3661383 0.71 RAB9A (0.57) RAB9ANPC1MAPTTP53SMN1; SMN2
SCHEMBL2108932 0.70 NPC1 (0.53) MCL1RAB9ANPC1MAPTATM
SCHEMBL3664746 0.70 HDAC4 (0.49) SMN1; SMN2LMNAFFAR1HDAC1HDAC4
SCHEMBL31036198 0.70 SMN1; SMN2 (0.72) MCL1RAB9ANPC1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP claimed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO claimed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP disclosed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO disclosed