SCHEMBL3661383

SCHEMBL3661383

O=C(O)Oc1nc(-c2ccccn2)no1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 12/20 0.57
NPC1 O15118 12/20 0.57
SMN1; SMN2 Q16637 11/20 0.57
PKM P14618 8/20 0.57
TP53 P04637 6/20 0.57
MAPT P10636 2/20 0.57
KMT2A Q03164 2/20 0.57
HTT P42858 1/20 0.54
ALDH1A1 P00352 5/20 0.52
TSHR P16473 3/20 0.52
KDM4E B2RXH2 3/20 0.52
HSD17B10 Q99714 2/20 0.52
LMNA P02545 1/20 0.52
HPGD P15428 1/20 0.52
KLF5 Q13887 1/20 0.52
GRM5 P41594 2/20 0.51
FAAH O00519 1/20 0.48
CES1 P23141 1/20 0.48
NCEH1 Q6PIU2 1/20 0.48
DAGLA Q9Y4D2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083201 0.80 NR1H4 (0.52) RAB9ANPC1SMN1; SMN2TP53MAPT
SCHEMBL493279 0.77 FAAH (0.61) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL2162094 0.73 NPC1 (0.54) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL4034138 0.73 NPC1 (0.65) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3666186 0.73 ALDH1A1 (0.43) RAB9ANPC1MAPTALDH1A1TSHR
SCHEMBL6384896 0.72 NPC1 (0.63) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL18078055 0.72 HTT (0.56) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL1424895 0.72 TP53 (0.77) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3517537 0.71 NPC1 (0.68) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3667161 0.71 ALDH1A1 (0.59) RAB9ANPC1SMN1; SMN2TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP claimed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO claimed
EP-2139851-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2010-01-06 EP disclosed
WO-2008131946-A2 SUBSTITUTED AMIDE DERIVATIVES Grünenthal GmbH (DE) 2008-11-06 WO disclosed