SCHEMBL4083201

SCHEMBL4083201

O=C(O)Oc1nc(-c2ccccc2)no1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.52
NOTUM Q6P988 2/20 0.49
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
ALDH1A1 P00352 2/20 0.48
CHUK O15111 1/20 0.46
CASP3 P42574 1/20 0.46
TXNRD1 Q16881 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
NOX4 Q9NPH5 1/20 0.46
GPR55 Q9Y2T6 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
TDP1 Q9NUW8 2/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
S1PR1 P21453 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27792725 0.87 NR1H4 (0.49) NR1H4NOTUMNPC1RAB9AALDH1A1
SCHEMBL3666056 0.82 KDM4E (0.54) NPC1RAB9AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL3664746 0.82 HDAC4 (0.49) CHUKTXNRD1NOX4SMN1; SMN2S1PR1
SCHEMBL3661383 0.80 RAB9A (0.57) NPC1RAB9AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL27766332 0.79 KMT2A (0.45) NOTUMALDH1A1SMN1; SMN2MAPK1MAPT
SCHEMBL3665206 0.79 DPP4 (0.43) NPC1RAB9AL3MBTL1S1PR1TSHR
SCHEMBL3666186 0.79 ALDH1A1 (0.43) NR1H4NPC1RAB9AALDH1A1TDP1
SCHEMBL27766331 0.78 KDM4E (0.50) ALDH1A1GAAMEN1KMT2A
SCHEMBL3661963 0.77 MAPT (0.59) NPC1RAB9AALDH1A1SMN1; SMN2MAPK1
SCHEMBL3667161 0.77 ALDH1A1 (0.59) NPC1RAB9AALDH1A1SMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2009520720-A 2009-05-28 JP claimed
EP-1989174-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2008-11-12 EP claimed
WO-2007079930-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO claimed
EP-2999469-A1 PHARMACEUTICAL COMPOSITION AND THE USE THEREOF, AND APPLICATION REGIME OF SAID PHARMACEUTICAL COMPOSITION FOR ON-DEMAND CONTRACEPTION Bayer Pharma Aktiengesellschaft (DE) 2016-03-30 EP disclosed
WO-2014187744-A1 PHARMACEUTICAL COMPOSITION AND THE USE THEREOF, AND APPLICATION REGIME OF SAID PHARMACEUTICAL COMPOSITION FOR ON-DEMAND CONTRACEPTION BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-11-27 WO disclosed
EP-1989174-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2008-11-12 EP disclosed
WO-2007079930-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO disclosed