SCHEMBL3665879

SCHEMBL3665879

CN(CCOc1cc(Br)ccc1NC(CO)N(C)Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
IKBKB O14920 1/20 0.42
KDM4E B2RXH2 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
TSHR P16473 1/20 0.40
ATM Q13315 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPC1 O15118 1/20 0.40
MCHR1 Q99705 1/20 0.39
CCR5 P51681 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1987646 0.74 LMNA (0.54) LMNAHTR1DHTR1BGAASMN1; SMN2
SCHEMBL3665876 0.74 LMNA (0.49) LMNAHTR1DHTR1BGAASMN1; SMN2
SCHEMBL3888894 0.71 LMNA (0.86) LMNAHTR1DHTR1BGAASMN1; SMN2
SCHEMBL1992407 0.70 LMNA (0.49) LMNAHTR1DHTR1BGAASMN1; SMN2
SCHEMBL6351462 0.65 AKR1C2 (0.58) SMN1; SMN2TSHRATMNPC1MCHR1
SCHEMBL781749 0.65 ADRA2B (0.46) LMNAGAAKDM4ETSHRATM
SCHEMBL8391031 0.65 HTR1D (0.63) LMNAHTR1DHTR1BTSHRATM
Hydrochloric Acid SCHEMBL8704830 0.64 HTR1D (0.62) LMNAHTR1DHTR1BTSHRATM
SCHEMBL8487152 0.64 HTR1D (0.62) LMNAHTR1DHTR1BSMN1; SMN2TSHR
SCHEMBL17682060 0.63 TSHR (0.81) HTR1DHTR1BKDM4ETSHRATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed