SCHEMBL3669304

SCHEMBL3669304

CNCCc1nc(-c2ccc(C(=O)O)cc2)c(C)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.54
RARG P13631 5/20 0.54
RARA P10276 4/20 0.54
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
POLB P06746 3/20 0.44
PKM P14618 2/20 0.44
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GAA P10253 2/20 0.43
MAPK1 P28482 1/20 0.43
ALDH1A1 P00352 5/20 0.42
MAPT P10636 1/20 0.42
OPRK1 P41145 1/20 0.42
PDE10A Q9Y233 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239090 0.75 RARA (0.68) RARBRARGRARAMEN1KMT2A
SCHEMBL3674507 0.75 CSNK2A1 (0.54) RARBRARGRARARAB9A
SCHEMBL1479736 0.73 RARA (0.57) RARBRARGRARAMEN1KMT2A
SCHEMBL1479738 0.73 RARA (0.57) RARBRARGRARAMEN1KMT2A
Hydrochloric Acid SCHEMBL5592169 0.72 RARA (0.56) RARBRARGRARAMEN1KMT2A
Hydrochloric Acid SCHEMBL5592171 0.72 RARA (0.56) RARBRARGRARAMEN1KMT2A
SCHEMBL9250705 0.71 ITGB3 (0.50) RARBRARGRARAMEN1KMT2A
SCHEMBL12876806 0.70 RARA (0.53) RARBRARGRARAMEN1KMT2A
SCHEMBL7481036 0.70 RARA (0.56) RARBRARGRARAMEN1KMT2A
Terephthalic Acid SCHEMBL11033093 0.69 TSHR (0.60) KMT2AMAPK1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2240491-A2 COMPOUNDS Amura Therapeutics Limited (GB) 2010-10-20 EP disclosed
WO-2009087379-A2 TETRAHYDROFURO (3, 2 -B) PYRROL- 3 -ONE DERIVATIVES AS INHIBITORS OF CYSTEINE PROTEINASES AMURA THERAPEUTICS LIMITED (GB) 2009-07-16 WO disclosed