SCHEMBL3671270

SCHEMBL3671270

CCOC(=O)C1CCN(c2ccccn2)C(N)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 4/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
TP53 P04637 1/20 0.44
ALOX12 P18054 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GAA P10253 1/20 0.44
LTA4H P09960 1/20 0.43
NPC1 O15118 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.43
NOS2 P35228 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2287525 0.86 CYP2C19 (0.47) CYP2C19ALDH1A1KDM4EKMT2AMEN1
SCHEMBL30745927 0.83 CYP2C19 (0.44) CYP2C19ALDH1A1KDM4EKMT2AMEN1
SCHEMBL5132804 0.83 CTSB (0.48) CYP2C19ALDH1A1KDM4EKMT2AMEN1
Hydrochloric Acid SCHEMBL30745936 0.82 CYP2C19 (0.44) CYP2C19ALDH1A1KDM4EKMT2AMEN1
SCHEMBL3352709 0.81 MAPT (0.57) CYP2C19ALDH1A1KDM4EKMT2AMEN1
SCHEMBL27775216 0.75 CYP2C19 (0.50) CYP2C19ALDH1A1KDM4EKMT2AMEN1
SCHEMBL3311153 0.75 KDM4E (0.46) ALDH1A1KDM4EKMT2AMAPTTP53
SCHEMBL9249018 0.73 NPC1 (0.42) ALDH1A1KDM4EMAPTTP53NPC1
SCHEMBL27673392 0.73 ALDH1A1 (0.55) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL2490913 0.73 DPP4 (0.47) ALDH1A1KDM4EMAPTTP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155687-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2010-02-24 EP disclosed
WO-2008141976-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS VIA PHARMACEUTICALS, INC. (US) 2008-11-27 WO disclosed