SCHEMBL9249018

SCHEMBL9249018

CCOC(=O)C1CC(O)CN1c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
CTSS P25774 1/20 0.41
ALDH1A1 P00352 5/20 0.41
NOS2 P35228 1/20 0.40
MAPT P10636 2/20 0.40
ATM Q13315 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRM1 Q13255 2/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
NPEPPS P55786 1/20 0.39
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251140 0.80 ITGB2 (0.48) GRM1ITGB2ICAM1ITGAL
SCHEMBL26255120 0.73 ALDH1A1 (0.47) NPC1TP53HPGDRAB9AALDH1A1
SCHEMBL3671270 0.73 CYP2C19 (0.47) NPC1TP53RAB9AALDH1A1NOS2
SCHEMBL2287525 0.73 CYP2C19 (0.47) NPC1TP53RAB9AALDH1A1NOS2
SCHEMBL4988396 0.72 NPEPPS (0.43) NPC1TP53HPGDRAB9AALDH1A1
SCHEMBL4984336 0.72 P2RX7 (0.42) NPC1TP53HPGDRAB9AALDH1A1
SCHEMBL28446474 0.72 NPC1 (0.41) NPC1TP53HPGDRAB9AALDH1A1
SCHEMBL5568192 0.72 MEN1 (0.50) ALDH1A1MAPTATMKDM4E
SCHEMBL8269795 0.72 MEN1 (0.50) ALDH1A1MAPTATMKDM4E
SCHEMBL4662072 0.72 MEN1 (0.50) ALDH1A1MAPTATMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405847-A Antiallergic, antiasthmatic, anxiolytic, hypotensive agents ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1995-04-11 US disclosed
CN-1088928-A New 4,5-dihydro-4-oxo-pyrrolo-[1,2-α] quinazolinone ASTA MEDICA AG (DE) 1994-07-06 CN disclosed
EP-0584487-A2 4,5-Dihydro-4-oxopyrrolo (1,2-a) quinoxalines and aza-analoges and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1994-03-02 EP disclosed