SCHEMBL3671907

SCHEMBL3671907

Cc1ccc(C)c(OCC2(C3(COc4c(Cl)cccc4Cl)NCCN3)NCCN2)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 2/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
RAB9A P51151 2/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTR1A P08908 3/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
SLC6A2 P23975 1/20 0.32
ADRA2A P08913 2/20 0.31
ADRA2B P18089 2/20 0.31
ADRA2C P18825 2/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
OPRK1 P41145 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3671905 0.72 HTR1D (0.55) HTR1AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL4630003 0.65 P2RX7 (0.36) POLBHTR1D
SCHEMBL3236165 0.63 RAB9A (0.50) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL12129099 0.62 KDM4E (0.62) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL27785923 0.61 KDM4E (0.56) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL6985548 0.60 NQO1 (0.42) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL1547567 0.60 L3MBTL1 (0.59) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL19122260 0.60 KDM4E (0.42) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL16572858 0.60 KDM4E (0.68) KDM4EKMT2AL3MBTL1RAB9AGAA
SCHEMBL14499037 0.60 SCN4A (0.61) KDM4EKMT2AL3MBTL1RAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173720-A2 2-IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. Hoffmann-Roche AG (CH) 2010-04-14 EP claimed
WO-2009003868-A2 2 -IMIDAZOLINES HAVING A GOOD AFFINITY TO THE TRACE AMINE ASSOCIATED RECEPTORS (TAARS) F. HOFFMANN-LA ROCHE AG (CH) 2009-01-08 WO claimed