SCHEMBL367330

SCHEMBL367330

CC(=O)c1ccc2c(C(N)=O)c3ccccc3n2c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.46
SRC P12931 2/20 0.46
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
NPC1 O15118 2/20 0.39
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
BAZ2B Q9UIF8 1/20 0.37
BAZ2A Q9UIF9 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367569 0.89 SRC (0.46) EGFRSRCALDH1A1HPGDKMT2A
SCHEMBL367764 0.89 EGFR (0.45) EGFRSRCALDH1A1HPGDNPC1
SCHEMBL366876 0.87 EGFR (0.44) EGFRSRCALDH1A1HPGDKMT2A
SCHEMBL365259 0.87 KDM4E (0.44) EGFRSRCALDH1A1HPGDHTR2A
Potassium Ion SCHEMBL364867 0.84 ALDH1A1 (0.40) EGFRSRCALDH1A1HPGDNPC1
SCHEMBL366442 0.83 ALDH1A1 (0.42) EGFRSRCALDH1A1HPGDNPC1
SCHEMBL364281 0.83 NR4A2 (0.48) EGFRSRCALDH1A1KMT2APOLB
SCHEMBL365635 0.82 IDO1 (0.44) EGFRSRCALDH1A1HPGDNPC1
SCHEMBL364389 0.82 ALDH1A1 (0.48) EGFRSRCALDH1A1HPGDNPC1
SCHEMBL366978 0.81 SCN9A (0.45) ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed