SCHEMBL3674076

SCHEMBL3674076

NC(=O)N(c1ccc(C(F)(F)F)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
KIF11 P52732 4/20 0.46
EPHX2 P34913 1/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
PLAU P00749 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
KMT2A Q03164 1/20 0.43
SRD5A2 P31213 1/20 0.42
GSK3B P49841 2/20 0.41
CYP1A2 P05177 1/20 0.41
PTPN1 P18031 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
PTGS1 P23219 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29624259 0.86 CES2 (0.47) CES2CES1KIF11EPHX2HTR3E
SCHEMBL21399416 0.83 CES2 (0.48) CES2CES1KIF11EPHX2HTR3E
SCHEMBL29727867 0.83 CYP3A4 (0.50) EPHX2
SCHEMBL28809584 0.80 CES2 (0.45) CES2CES1KIF11EPHX2HTR3E
SCHEMBL525760 0.80 CES2 (0.45) CES2CES1KIF11EPHX2HTR3E
SCHEMBL8405808 0.80 KIF11 (0.44) CES2CES1KIF11EPHX2HTR3E
SCHEMBL11022026 0.79 CASP1 (0.40) CES2CES1KIF11EPHX2KMT2A
SCHEMBL2717803 0.79 ALDH1A1 (0.46) KIF11EPHX2KMT2ASRD5A2CYP1A2
SCHEMBL16345980 0.79 CES2 (0.48) CES2
SCHEMBL31188158 0.78 TACR1 (0.49) CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150056160-A1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA TEXAS PHARMACEUTICALS, INC. 2015-02-26 US claimed
EP-1098641-B1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA ST JUDE PHARMACEUTICALS INC (US) 2016-04-27 EP disclosed
US-20150056160-A1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA TEXAS PHARMACEUTICALS, INC. 2015-02-26 US disclosed
US-20100056643-A1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA ST. JUDE PHARMACEUTICALS, INC. 2010-03-04 US disclosed
US-7635722-B1 Chemical induced intracellular hyperthermia Saint Jude Pharmaceuticals, Inc. (US) 2009-12-22 US disclosed