SCHEMBL3683993

SCHEMBL3683993

O=C(c1nc2c(C(F)(F)F)cc(-c3ccco3)cn2c1Cl)N1CCCC(c2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
SCD5 Q86SK9 5/20 0.48
CACNA1B Q00975 1/20 0.45
APBA1 Q02410 1/20 0.45
RAB9A P51151 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SCD O00767 1/20 0.42
HSD11B1 P28845 1/20 0.42
PROKR1 Q8TCW9 2/20 0.41
RHOA P61586 1/20 0.41
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
SCN9A Q15858 1/20 0.40
PTPN7 P35236 1/20 0.40
DUSP3 P51452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3687507 0.96 SCD5 (0.53) ALDH1A1SCD5CACNA1BAPBA1RAB9A
SCHEMBL3689454 0.92 SCD5 (0.47) ALDH1A1SCD5CACNA1BAPBA1RAB9A
SCHEMBL3694395 0.90 SCD5 (0.45) ALDH1A1SCD5CACNA1BAPBA1RAB9A
SCHEMBL3690897 0.88 ALDH1A1 (0.46) ALDH1A1RAB9ATDP1L3MBTL1LMNA
SCHEMBL3691708 0.86 SCD (0.45) SCD5SCD
SCHEMBL3693859 0.86 P2RX7 (0.43) ALDH1A1SCD5CACNA1BAPBA1RAB9A
SCHEMBL3690063 0.84 SCD5 (0.45) ALDH1A1SCD5SCDLMNAMAPT
SCHEMBL3689489 0.83 MAPT (0.51) ALDH1A1SCD5RAB9AL3MBTL1SCD
SCHEMBL3691242 0.83 SCD5 (0.48) SCD5CACNA1BAPBA1RAB9ASCD
SCHEMBL3692964 0.83 SCD5 (0.48) SCD5CACNA1BAPBA1RAB9ASCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
EP-2187883-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2010-05-26 EP disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed
WO-2009023179-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2009-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections OAT, HAVCR2, CPS1 ALDH1A1 1337/4885SCD5 2314/4885CACNA1B 1940/4885
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections OAT, HAVCR2, CPS1 ALDH1A1 1337/4885SCD5 2314/4885CACNA1B 1940/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.