SCHEMBL3684483

SCHEMBL3684483

CN(C)Cc1cccc(C(=O)C=Cc2cc(N3CCN(C)CC3)ccc2-c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 10/20 0.49
HDAC4 P56524 10/20 0.49
HDAC1 Q13547 10/20 0.49
HDAC7 Q8WUI4 10/20 0.49
HDAC2 Q92769 10/20 0.49
HDAC10 Q969S8 10/20 0.49
HDAC11 Q96DB2 10/20 0.49
HDAC8 Q9BY41 10/20 0.49
HDAC6 Q9UBN7 10/20 0.49
HDAC9 Q9UKV0 10/20 0.49
HDAC5 Q9UQL6 10/20 0.49
BCHE P06276 1/20 0.46
AOC3 Q16853 2/20 0.44
HTR6 P50406 1/20 0.42
HTR2C P28335 2/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
DRD1 P21728 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686624 0.85 PTPN1 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3694114 0.85 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3688795 0.85 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3696557 0.84 HDAC3 (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3684481 0.81 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3688945 0.81 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3685240 0.81 CTSL (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3690600 0.81 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3686024 0.81 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3687288 0.78 BCHE (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed