SCHEMBL3686624

SCHEMBL3686624

COc1ccc(C(=O)C=Cc2cc(N3CCN(C)CC3)ccc2-c2ccccc2)cc1CN(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.44
KEAP1 Q14145 2/20 0.43
NFE2L2 Q16236 2/20 0.43
HSP90AA1 P07900 1/20 0.43
DNMT1 P26358 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
TNNI3 P19429 1/20 0.42
TNNT2 P45379 1/20 0.42
TNNC1 P63316 1/20 0.42
HDAC3 O15379 4/20 0.42
HDAC4 P56524 4/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC7 Q8WUI4 4/20 0.42
HDAC2 Q92769 4/20 0.42
HDAC10 Q969S8 4/20 0.42
HDAC11 Q96DB2 4/20 0.42
HDAC8 Q9BY41 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3684483 0.85 HDAC3 (0.49) PTPN1MAPTHDAC3HDAC4HDAC1
SCHEMBL3688874 0.83 ABCB1 (0.45) MEN1KMT2AMAPTHDAC3HDAC4
SCHEMBL3686623 0.83 ABCB1 (0.45) MEN1KMT2AMAPTHDAC3HDAC4
SCHEMBL3686880 0.81 KEAP1 (0.43) PTPN1KEAP1NFE2L2HSP90AA1DNMT1
SCHEMBL3685240 0.80 CTSL (0.53) PTPN1HSP90AA1MEN1KMT2AMAPT
SCHEMBL3688723 0.80 KEAP1 (0.43) KEAP1NFE2L2MEN1KMT2AMAPT
SCHEMBL3687122 0.80 KEAP1 (0.43) KEAP1NFE2L2MEN1KMT2AMAPT
SCHEMBL3686504 0.79 HSP90AA1 (0.41) KEAP1NFE2L2HSP90AA1DNMT1MEN1
SCHEMBL3696557 0.77 HDAC3 (0.47) PTPN1HDAC3HDAC4HDAC1HDAC7
SCHEMBL5915509 0.77 HSP90AA1 (0.57) PTPN1HSP90AA1DNMT1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP claimed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed