Indene

Indene

SCHEMBL368620

C1=Cc2ccccc2C1.C=C(C)c1ccccc1

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.72
CYP2C19 P33261 1/20 0.72
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
HSD17B3 P37058 1/20 0.33
CES2 O00748 2/20 0.32
CES1 P23141 2/20 0.32
PARP1 P09874 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
XBP1 P17861 1/20 0.30
ATM Q13315 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indene SCHEMBL28692932 0.87 CYP2D6 (0.56) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL28841652 0.87 CYP2D6 (0.56) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL10603166 0.85 CYP2D6 (0.57) CYP2D6CYP2C19CA1CA2
Indene SCHEMBL2769732 0.83 CYP2D6 (0.53) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL5689989 0.83 CYP2D6 (0.53) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL29746662 0.82 CYP2D6 (0.51) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL89373 0.82 CYP2D6 (0.51) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL8662549 0.82 CYP2C19 (0.53) CYP2D6CYP2C19CA1CA2LMNA
Indene SCHEMBL7745309 0.81 CYP2D6 (0.50) CYP2D6CYP2C19CA1CA2HSD17B3
Indene SCHEMBL28216169 0.81 CA1 (0.50) CYP2D6CYP2C19CA1CA2HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3581398-B1 RUBBER COMPOSITION FOR TIRE, AND PNEUMATIC TIRE SUMITOMO RUBBER IND (JP) 2020-09-16 EP claimed
CN-103946299-B Rubber composition and pneumatic tire 住友橡胶工业株式会社 2018-10-09 CN disclosed
CN-103946302-B Rubber composition and pneumatic tire 住友橡胶工业株式会社 2018-05-15 CN disclosed
EP-2772514-B1 RUBBER COMPOSITION, AND PNEUMATIC TIRE SUMITOMO RUBBER IND (JP) 2017-08-16 EP disclosed
US-9428641-B2 Rubber composition, and pneumatic tire SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2016-08-30 US disclosed
EP-2749594-B1 RUBBER COMPOSITION AND STUDLESS TIRE SUMITOMO RUBBER IND (JP) 2016-06-08 EP disclosed
EP-2772511-B1 RUBBER COMPOSITION, AND PNEUMATIC TIRE SUMITOMO RUBBER IND (JP) 2016-06-08 EP disclosed
US-9290644-B2 Rubber composition, and pneumatic tire SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2016-03-22 US disclosed
US-20140296376-A1 RUBBER COMPOSITION, AND PNEUMATIC TIRE SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2014-10-02 US disclosed
US-20140256847-A1 RUBBER COMPOSITION, AND PNEUMATIC TIRE SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2014-09-11 US disclosed
EP-2772514-A1 RUBBER COMPOSITION, AND PNEUMATIC TIRE Sumitomo Rubber Industries, Ltd. (JP) 2014-09-03 EP disclosed
EP-2772511-A1 RUBBER COMPOSITION, AND PNEUMATIC TIRE Sumitomo Rubber Industries, Ltd. (JP) 2014-09-03 EP disclosed
US-20140213693-A1 RUBBER COMPOSITION AND STUDLESS TIRE SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2014-07-31 US disclosed
EP-2749594-A1 RUBBER COMPOSITION AND STUDLESS TIRE Sumitomo Rubber Industries, Ltd. (JP) 2014-07-02 EP disclosed
US-8318861-B2 Rubber composition and tire using the same BRIDGESTONE CORPORATION (JP) 2012-11-27 US disclosed
EP-2103650-B1 RUBBER COMPOSITION AND TIRE USING THE SAME BRIDGESTONE CORP (JP) 2012-08-08 EP disclosed
US-20120016056-A1 RUBBER COMPOSITION FOR TREAD AND PNEUMATIC TIRE SUMITOMO RUBBER INDUSTRIES, LTD. (JP) 2012-01-19 US disclosed
US-20100113703-A1 RUBBER COMPOSITION AND TIRE USING THE SAME BRIDGESTONE CORPORATION (JP) 2010-05-06 US disclosed
EP-2103650-A1 RUBBER COMPOSITION AND TIRE USING THE SAME Bridgestone Corporation (JP) 2009-09-23 EP disclosed