SCHEMBL3687356

SCHEMBL3687356

O=C(c1nc2c(C(F)(F)F)cc(Br)cn2c1Br)N1CCC(c2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD5 Q86SK9 6/20 0.50
RAB9A P51151 5/20 0.44
NPC1 O15118 4/20 0.44
ATM Q13315 1/20 0.44
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
SCD O00767 2/20 0.42
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SPR P35270 1/20 0.40
SCN9A Q15858 1/20 0.40
TSHR P16473 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649698 0.92 RAB9A (0.43) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3687818 0.86 SCD5 (0.47) SCD5RAB9ANPC1ATMMAPT
SCHEMBL7496545 0.86 RAB9A (0.47) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3683970 0.85 ROCK2 (0.51) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3688270 0.84 SCD5 (0.51) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3689754 0.83 NPC1 (0.42) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3688733 0.82 SCD5 (0.47) SCD5RAB9ANPC1ATM
SCHEMBL3689413 0.78 SCD5 (0.38) SCD5RAB9ANPC1ATMMAPT
SCHEMBL3691914 0.78 SCD5 (0.44) SCD5RAB9ANPC1ATMSCD
SCHEMBL3696196 0.77 ROCK2 (0.43) SCD5RAB9ANPC1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections GLAXOSMITHKLINE LLC 2012-05-17 US disclosed
EP-2187883-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2010-05-26 EP disclosed
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections GLAXOSMITHKLINE LLC 2009-07-09 US disclosed
WO-2009023179-A2 NITROGEN CONTAINING BICYCLIC CHEMICAL ENTITIES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2009-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121540-A1 Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections OAT, HAVCR2, CPS1 SCD5 2314/4885RAB9A 3638/4885NPC1 229/4885
US-20090176778-A1 Certain nitrogen containing bicyclic chemical entities for treating viral infections OAT, HAVCR2, CPS1 SCD5 2314/4885RAB9A 3638/4885NPC1 229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.