SCHEMBL3698321

SCHEMBL3698321

COc1cccc2c(C(CO)N3C4CCC3CC(NCc3cc5ccccc5o3)C4)ccnc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
HTR2B P41595 6/20 0.35
DRD2 P14416 5/20 0.35
HTR1A P08908 4/20 0.35
CYP3A4 P08684 1/20 0.34
HTR3A P46098 1/20 0.34
KCNH2 Q12809 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
CCR8 P51685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690604 0.86 SLC2A1 (0.36) HCRTR1HCRTR2HTR2BDRD2HTR1A
SCHEMBL5652075 0.85 CCR8 (0.45) HTR2BDRD2CYP3A4KCNH2KDM4E
SCHEMBL5777778 0.80 SLC2A1 (0.47) HTR2BDRD2HTR1ACYP3A4KCNH2
SCHEMBL3688489 0.76 HTR1A (0.33) HTR1AMEN1ALDH1A1KMT2AADRA1D
SCHEMBL3687758 0.72 CNR2 (0.33) HTR1ACYP2C19ADRA1DADRA1AADRA1B
SCHEMBL3690599 0.71 KCNH2 (0.50) CYP3A4KCNH2KDM4EMEN1ALDH1A1
SCHEMBL5778069 0.71 MEN1 (0.38) HTR2BDRD2HTR1ACYP3A4KCNH2
SCHEMBL3694994 0.69
SCHEMBL4275508 0.65 KCNH2 (0.65) KCNH2CCR8
SCHEMBL3697149 0.64 HTR1A (0.35) HTR2BHTR1AALDH1A1ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed