SCHEMBL3689290

SCHEMBL3689290

CN1CCN(c2cc(C=O)cc(-c3ccccc3)c2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
HTR3A P46098 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
MELK Q14680 1/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
KIF11 P52732 2/20 0.41
ADRA2C P18825 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.40
MAPKAPK2 P49137 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696108 0.83 ALDH1A1 (0.50) ALDH1A1HTR3AMAPK1ADRA2CTSHR
SCHEMBL3686236 0.79 ALDH1A1 (0.46) ALDH1A1MAPK1TSHR
SCHEMBL3690173 0.76 ALDH1A1 (0.59) ALDH1A1HTR3ASMN1; SMN2MAPTMAPK1
SCHEMBL29442412 0.76 ALDH1A1 (0.64) ALDH1A1HTR3AMAPTMAPK1ADRA2C
SCHEMBL1444185 0.76 ALDH1A1 (0.64) ALDH1A1HTR3AMAPTMAPK1ADRA2C
SCHEMBL30108214 0.76 HTR1A (0.64) ALDH1A1HTR3ASMN1; SMN2MAPK1ADRA2C
SCHEMBL22579268 0.74 ALDH1A1 (0.89) ALDH1A1SMN1; SMN2MAPTMAOAMAOB
SCHEMBL30108226 0.73 MELK (0.60) ALDH1A1HTR3ASMN1; SMN2NPC1MAPT
SCHEMBL1664238 0.73 ALDH1A1 (0.55) ALDH1A1NPC1MAPTRAB9APOLB
SCHEMBL7902633 0.73 ALDH1A1 (0.55) ALDH1A1NPC1MAPTRAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed