SCHEMBL3690489

SCHEMBL3690489

CC(C)(C)C(Cc1cc(-c2cccnc2F)c(S(=O)(=O)c2ncc[nH]2)s1)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 18/20 0.35
CYP3A4 P08684 1/20 0.34
DYRK1A Q13627 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3703109 0.95 AGTR2 (0.33) AGTR2CYP3A4
SCHEMBL3654949 0.85 AGTR2 (0.33) AGTR2CYP3A4
SCHEMBL3649952 0.85 ABCC9 (0.36) AGTR2KMT2A
SCHEMBL3804718 0.84 ABCC9 (0.36) AGTR2CYP3A4
SCHEMBL3652361 0.83 AGTR2 (0.33) AGTR2CYP3A4DYRK1A
SCHEMBL3806158 0.83 AGTR2 (0.32) AGTR2CYP3A4
SCHEMBL3803071 0.82 KDM4E (0.33) AGTR2KMT2A
Hydrochloric Acid SCHEMBL3645134 0.82 NAMPT (0.33) AGTR2KMT2A
SCHEMBL4028250 0.81 AGTR2 (0.32) AGTR2CYP3A4
SCHEMBL4125945 0.81 LIPG (0.33) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed