SCHEMBL369133

SCHEMBL369133

Clc1nc2cccnc2s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.58
NPC1 O15118 10/20 0.53
RAB9A P51151 9/20 0.53
SMN1; SMN2 Q16637 5/20 0.53
POLB P06746 2/20 0.50
ATM Q13315 1/20 0.42
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 8/20 0.41
MAPT P10636 4/20 0.41
HPGD P15428 4/20 0.41
GAA P10253 3/20 0.41
RUNX1 Q01196 3/20 0.41
CBFB Q13951 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
ALOX12 P18054 1/20 0.41
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30775052 1.00 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
Hydrochloric Acid SCHEMBL1896253 0.98 PDK1 (0.56) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL30190003 0.77 PDK1 (0.60) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL140126 0.77 PDK1 (0.60) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL137507 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL13310867 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL2642887 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL15689525 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL1761326 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL2176039 0.75 PDK1 (0.58) PDK1NPC1RAB9ASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4634170-A1 IMIDAZO[4,5-B]PYRIDINE DERIVATIVES AS PCSK9 INHIBITORS AND METHODS OF USE THEREOF AstraZeneca AB (SE) 2025-10-22 EP disclosed
US-20250197387-A1 BCL-XL DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-06-19 US disclosed
EP-3676261-B1 SUBSTITUTED 2-AZABICYCLO[3.1.1]HEPTANE AND 2-AZABICYCLO[3.2.1]OCTANE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS CHRONOS THERAPEUTICS LTD (GB) 2024-12-18 EP disclosed
EP-4401729-A1 BCL-XL DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2024-07-24 EP disclosed
US-20240239767-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2024-07-18 US disclosed
WO-2024126773-A1 IMIDAZO[4,5-B]PYRIDINE DERIVATIVES AS PCSK9 INHIBITORS AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2024-06-20 WO disclosed
WO-2023229380-A1 HETEROCYCLIC COMPOUND AS DIACYLGLYCEROL KINASE INHIBITOR AND USE THEREOF 주식회사 엘지화학 2023-11-30 WO disclosed
US-11660293-B2 Substituted 2-azabicyclo[3.1.1]heptane and 2-azabicyclo[3.2.1]octane derivatives as orexin receptor antagonists CHRONOS THERAPEUTICS LIMITED (GB) 2023-05-30 US disclosed
US-11660293-B2 Substituted 2-azabicyclo[3.1.1]heptane and 2-azabicyclo[3.2.1]octane derivatives as orexin receptor antagonists CHRONOS THERAPEUTICS LIMITED (GB) 2023-05-30 US disclosed
US-11660293-B2 Substituted 2-azabicyclo[3.1.1]heptane and 2-azabicyclo[3.2.1]octane derivatives as orexin receptor antagonists CHRONOS THERAPEUTICS LIMITED (GB) 2023-05-30 US disclosed
US-20070265298-A1 Preparation and Use of Biphenyl-4-Yl-Carbonylamino Acid Derivatives for the Treatment of Obesity BAYER PHARMACEUTICALS CORPORATION (US) 2007-11-15 US disclosed
US-20050112770-A1 Method for optical measurement of multi-stranded nucleic acid FUJI PHOTO FILM CO., LTD. 2005-05-26 US disclosed
EP-1362894-A2 Method for optical measurement of multi-stranded nucleic acid using cyanine dyes FUJI PHOTO FILM CO., LTD. (JP) 2003-11-19 EP disclosed
US-5616717-A Process for the preparation of pure enantiomers of 1-(2-pyridyl)-2-cyclohexylethylamine BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-04-01 US disclosed
US-5552421-A Leukotriene biosynthesis inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1996-09-03 US disclosed
US-5374644-A Insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-12-20 US disclosed
US-5296486-A Leukotriene biosynthesis inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1994-03-22 US disclosed
EP-0535521-A2 Condensed oxazole and thiazole derivatives as leukotriene biosynthesis inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1993-04-07 EP disclosed
EP-0256667-B1 SUBSTITUTED PHENYL-2-PROPENOIC ACID DERIVATIVES USEFUL IN AGRICULTURE IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-12-30 EP disclosed
EP-0256667-A2 Substituted phenyl-2-propenoic acid derivatives useful in agriculture IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-02-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070265298-A1 Preparation and Use of Biphenyl-4-Yl-Carbonylamino Acid Derivatives for the Treatment of Obesity FABP4, GPR119, PGC PDK1 291/4885NPC1 466/4885RAB9A 2219/4885
US-20240239767-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF PCSK9, PCSK7, PCSK6 PDK1 3666/4885NPC1 100/4885RAB9A 1724/4885
US-20250197387-A1 BCL-XL DEGRADERS AND USES THEREOF XIAP, BCL2L1, BCL2L10 PDK1 1837/4885NPC1 4285/4885RAB9A 1966/4885
US-11660293-B2 Substituted 2-azabicyclo[3.1.1]heptane and 2-azabicyclo[3.2.1]octane derivatives as orexin receptor antagonists HCRTR2, HCRTR1, NPY1R PDK1 1614/4885NPC1 492/4885RAB9A 2293/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.