Berberine

Berberine

SCHEMBL3691964

CCO.COc1ccc2cc3[n+](cc2c1OC)CCc1cc2c(cc1-3)OCO2

nearest known ligand 0.90

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Known targets — ChEMBL curated mechanism

MMP1MMP13MMP7MMP8polrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Berberine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 8/20 0.90
ACHE P22303 8/20 0.90
EP300 Q09472 4/20 0.90
ALDH1A1 P00352 2/20 0.90
LMNA P02545 2/20 0.90
CYP3A4 P08684 2/20 0.90
CYP2D6 P10635 2/20 0.90
MAPT P10636 2/20 0.90
CHRM1 P11229 2/20 0.90
DRD2 P14416 2/20 0.90
TSHR P16473 2/20 0.90
ADRA2B P18089 2/20 0.90
ADRA2C P18825 2/20 0.90
RXRA P19793 2/20 0.90
DRD1 P21728 2/20 0.90
HTR2B P41595 2/20 0.90
HTT P42858 2/20 0.90
RAD52 P43351 2/20 0.90
KCNH2 Q12809 2/20 0.90
SMN1; SMN2 Q16637 2/20 0.90

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Berberine SCHEMBL25632 0.95 ACHE (1.00) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL15669190 0.95 ACHE (1.00) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL30153843 0.95 ACHE (1.00) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL29354144 0.95 ACHE (1.00) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL2538316 0.94 ACHE (0.98) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL4894622 0.94 BCHE (0.98) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL3686644 0.94 ACHE (0.98) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL21462194 0.94 ACHE (0.98) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL153906 0.94 ACHE (1.00) BCHEACHEEP300ALDH1A1LMNA
Berberine SCHEMBL10709599 0.94 ACHE (0.98) BCHEACHEEP300ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100292178-A1 Method of treating non-insulin dependent diabetes mellitus and related complications YOUNG JEFFREY 2010-11-18 US disclosed
US-20050019435-A1 Method of treating non-insulin dependent diabetes mellitus and related complications YOUNG JEFFREY (US) 2005-01-27 US disclosed