SCHEMBL3695443

SCHEMBL3695443

CN(C)CCN(C)c1cc(Br)cc(C=O)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
ALDH1A3 P47895 3/20 0.33
ALDH3A1 P30838 2/20 0.33
CYP2A6 P11509 1/20 0.32
CYP2A13 Q16696 1/20 0.32
TAAR1 Q96RJ0 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686497 0.75 ALDH1A1 (0.40) ALDH1A1ALDH1A3ALDH3A1CYP2A6CYP2A13
SCHEMBL3689253 0.73 CYP2A6 (0.57) ALDH1A1ALDH1A3ALDH3A1CYP2A6CYP2A13
SCHEMBL3688543 0.71 HTR7 (0.44) ALDH1A1KDM4E
SCHEMBL6121307 0.70 LMNA (0.41) ALDH1A1ALDH1A3ALDH3A1CYP2A6CYP2A13
SCHEMBL3689552 0.69 FLT3 (0.39) ALDH1A1KDM4EMEN1CYP1A2CYP2D6
SCHEMBL646947 0.69 ALDH1A1 (0.56) ALDH1A1ALDH1A3CYP2A6KDM4E
SCHEMBL708554 0.69 ALDH1A1 (0.56) ALDH1A1ALDH1A3CYP2A6KDM4E
SCHEMBL15008733 0.68 TAAR1 (0.55) ALDH1A1TAAR1KDM4EKMT2A
SCHEMBL21115197 0.66 TAAR1 (0.54) ALDH1A1CYP2A6TAAR1KDM4ECYP2D6
SCHEMBL13645995 0.66 CYP2A6 (0.64) ALDH1A1ALDH1A3ALDH3A1CYP2A6CYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed