SCHEMBL3689552

SCHEMBL3689552

CN(C)CCCNc1cc(Br)cc(C=O)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 5/20 0.39
KDM4E B2RXH2 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ALDH1A1 P00352 2/20 0.37
EGFR P00533 2/20 0.35
DRD3 P35462 1/20 0.35
APAF1 O14727 1/20 0.35
RAD52 P43351 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35
CASP8 Q14790 1/20 0.35
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
KMT2A Q03164 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5736369 0.76 LMNA (0.43) FLT3KDM4EL3MBTL1ALDH1A1DRD3
SCHEMBL3690875 0.74 HTR7 (0.40) FLT3KDM4EL3MBTL1DRD3APAF1
SCHEMBL3690211 0.72 MAOB (0.37) KDM4EL3MBTL1ALDH1A1
SCHEMBL2532889 0.72 ACHE (0.43) FLT3KDM4EALDH1A1DRD3CYP1A2
SCHEMBL24568765 0.71 KDR (0.46) FLT3KDM4EL3MBTL1EGFRRAD52
SCHEMBL21541819 0.71 TAAR1 (0.47) FLT3KDM4EL3MBTL1ALDH1A1EGFR
SCHEMBL3695443 0.69 ALDH1A1 (0.35) KDM4EALDH1A1MEN1CYP1A2CYP2D6
SCHEMBL15301101 0.68 NOS2 (0.45) FLT3EGFRCYP1A2
SCHEMBL2278503 0.68 HTR7 (0.46) ALDH1A1RAD52CYP1A2CYP2D6
SCHEMBL31453711 0.67 L3MBTL1 (0.44) FLT3KDM4EL3MBTL1DRD3APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed