Bicarbonate

Bicarbonate

SCHEMBL3696258

CC(C(C(=O)Nc1cccc(CC2CC2)c1)c1ccc(Cn2nc(C(F)(F)F)ccc2=O)cc1)C(F)(F)F.O=C(O)O

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNJ6 P48051 3/20 0.39
KCNJ5 P48544 3/20 0.39
KCNJ3 P48549 3/20 0.39
ACKR3 P25106 6/20 0.37
MET P08581 3/20 0.37
CCR3 P51677 1/20 0.37
KLKB1 P03952 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1178248 0.88 KCNJ6 (0.39) KCNJ6KCNJ5KCNJ3ACKR3MET
SCHEMBL1178051 0.88 KCNJ6 (0.40) KCNJ6KCNJ5KCNJ3MET
SCHEMBL3699959 0.88 KCNJ6 (0.42) KCNJ6KCNJ5KCNJ3MET
SCHEMBL7601286 0.86 KCNJ6 (0.39) KCNJ6KCNJ5KCNJ3ACKR3MET
SCHEMBL7601160 0.86 KCNJ6 (0.38) KCNJ6KCNJ5KCNJ3ACKR3MET
Bicarbonate SCHEMBL3692775 0.85 PTGES (0.45) ACKR3CCR3KLKB1
SCHEMBL1178386 0.85 MET (0.41) KCNJ6KCNJ5KCNJ3ACKR3MET
SCHEMBL1178284 0.82 MET (0.38) KCNJ6KCNJ5KCNJ3ACKR3MET
Bicarbonate SCHEMBL16735564 0.82 ACKR3 (0.47) ACKR3CCR3
Bicarbonate SCHEMBL9900300 0.82 ALDH1A1 (0.43) KCNJ6KCNJ5KCNJ3ACKR3CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed