SCHEMBL3698417

SCHEMBL3698417

CC(C)(C)C(Cc1cc(S(=O)(=O)c2ccccc2)n(-c2cccnc2C#N)n1)NC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLCG1 P19174 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ABCC9 O60706 2/20 0.32
ABCC8 Q09428 2/20 0.32
KCNJ11 Q14654 2/20 0.32
KCNJ8 Q15842 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
CYP2C9 P11712 1/20 0.31
NAMPT P43490 1/20 0.31
SLC5A1 P13866 1/20 0.30
P2RX7 Q99572 2/20 0.30
CNR1 P21554 1/20 0.30
HTR6 P50406 1/20 0.30
KCNH2 Q12809 1/20 0.30
SLC16A3 O15427 1/20 0.30
SLC16A1 P53985 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696124 0.95 CNR1 (0.31) PLCG1PTGDR2SLC5A1P2RX7CNR1
SCHEMBL3700741 0.87 PTGDR2 (0.34) MEN1KMT2ANPC1RAB9AABCC9
SCHEMBL3697760 0.85 NR1I2 (0.35) MEN1KMT2ANPC1RAB9AABCC9
SCHEMBL476393 0.84 APLNR (0.34) NAMPT
SCHEMBL476324 0.82 COMT (0.35) PTGDR2P2RX7HTR6KCNH2
SCHEMBL3697998 0.81 P2RX7 (0.35) MEN1KMT2ANPC1RAB9AABCC9
SCHEMBL3697138 0.81 SLC16A3 (0.34) MEN1KMT2AABCC9ABCC8KCNJ11
SCHEMBL476413 0.81 ABCC9 (0.35) ABCC9ABCC8KCNJ11KCNJ8NAMPT
SCHEMBL4137769 0.81 HTT (0.36) PTGDR2CYP2C9NAMPTP2RX7CNR1
SCHEMBL3701582 0.80 SLC16A3 (0.38) MEN1KMT2ANAMPTCNR1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed