SCHEMBL3698418

SCHEMBL3698418

CC(C)(C)CN(Cc1cc(S(=O)(=O)c2ccccc2)n(-c2cccnc2C#N)n1)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.32
CTSK P43235 2/20 0.32
PLCG1 P19174 1/20 0.31
P2RX7 Q99572 1/20 0.31
SLC16A3 O15427 1/20 0.30
SLC16A1 P53985 1/20 0.30
ABCC9 O60706 2/20 0.30
ABCC8 Q09428 2/20 0.30
KCNJ11 Q14654 2/20 0.30
KCNJ8 Q15842 2/20 0.30
ELANE P08246 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696127 0.95 P2RX7 (0.32) PTGDR2P2RX7SLC16A3SLC16A1
SCHEMBL3700744 0.88 PTGDR2 (0.33) PTGDR2SLC16A3SLC16A1ABCC9ABCC8
SCHEMBL4137765 0.87 NAMPT (0.33) PTGDR2P2RX7SLC16A3SLC16A1ELANE
SCHEMBL3697762 0.85 KDM4E (0.33) PTGDR2P2RX7SLC16A3SLC16A1ABCC9
SCHEMBL476395 0.84 NAMPT (0.33)
SCHEMBL3698416 0.83 HTR2C (0.42) PTGDR2PLCG1SLC16A3SLC16A1MEN1
SCHEMBL476326 0.82 COMT (0.36) PTGDR2KMT2A
SCHEMBL3697999 0.82 P2RX7 (0.33) PTGDR2P2RX7SLC16A3SLC16A1ABCC9
SCHEMBL3697140 0.80 SLC16A3 (0.34) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL476415 0.80 HTR6 (0.35) SLC16A3SLC16A1ABCC9ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed