SCHEMBL3700744

SCHEMBL3700744

CC(C)(C)CN(Cc1cc(S(=O)(=O)c2ccccc2)n(-c2cccnc2F)n1)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.33
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
NPSR1 Q6W5P4 2/20 0.33
SLC16A3 O15427 4/20 0.32
SLC16A1 P53985 4/20 0.32
ABCC9 O60706 3/20 0.32
ABCC8 Q09428 3/20 0.32
KCNJ11 Q14654 3/20 0.32
KCNJ8 Q15842 3/20 0.32
HTR6 P50406 4/20 0.32
POLB P06746 2/20 0.31
KDM4E B2RXH2 1/20 0.31
COMT P21964 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL476326 0.95 COMT (0.36) PTGDR2KMT2AHTR6KDM4ECOMT
SCHEMBL3697999 0.93 P2RX7 (0.33) PTGDR2ALDH1A1SLC16A3SLC16A1ABCC9
SCHEMBL476415 0.92 HTR6 (0.35) ALDH1A1MEN1KMT2ASLC16A3SLC16A1
SCHEMBL476339 0.91 HTR6 (0.32) HTR6
SCHEMBL3705969 0.90 SLC16A3 (0.39) PTGDR2SLC16A3SLC16A1ABCC9ABCC8
SCHEMBL476395 0.89 NAMPT (0.33)
SCHEMBL3697762 0.88 KDM4E (0.33) PTGDR2ALDH1A1SLC16A3SLC16A1ABCC9
SCHEMBL3698418 0.88 PTGDR2 (0.32) PTGDR2MEN1KMT2ASLC16A3SLC16A1
SCHEMBL3697140 0.87 SLC16A3 (0.34) KMT2ASLC16A3SLC16A1ABCC9ABCC8
SCHEMBL3808574 0.86 ABCC9 (0.35) ALDH1A1SLC16A3SLC16A1ABCC9ABCC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed