SCHEMBL370010

SCHEMBL370010

Cc1ccccc1C(CC(=O)c1ccc(=O)[nH]c1)c1ccc(C2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 5/20 0.44
NAMPT P43490 1/20 0.43
TRPV6 Q9H1D0 1/20 0.41
KDM4E B2RXH2 2/20 0.39
THRB P10828 2/20 0.39
MAPT P10636 2/20 0.39
PKM P14618 1/20 0.39
HPGDS O60760 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
NPC1L1 Q9UHC9 1/20 0.38
USP30 Q70CQ3 1/20 0.37
TP53 P04637 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
P2RY14 Q15391 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370011 1.00 GPR119 (0.44) GPR119NAMPTTRPV6KDM4ETHRB
SCHEMBL369411 0.89 TRPV6 (0.45) TRPV6MEN1KMT2AGAA
SCHEMBL368537 0.85 NAMPT (0.43) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL368536 0.85 NAMPT (0.43) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL14936621 0.84 NAMPT (0.44) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL1390947 0.83 GPR119 (0.46) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL14965873 0.83 NAMPT (0.42) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL363900 0.83 GPR119 (0.46) GPR119NAMPTKDM4ETHRBMAPT
SCHEMBL368574 0.82 GPBAR1 (0.51) GPR119NAMPTKDM4ETHRBPKM
SCHEMBL368575 0.82 GPBAR1 (0.51) GPR119NAMPTKDM4ETHRBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed
US-8765730-B2 1-hydroxyimino-3-phenyl-propanes Hoffmann-La Roche Inc (US) 2014-07-01 US disclosed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed
US-20120010190-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010190-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES GPBAR1, GPR119, ADRB1 GPR119 2/4885NAMPT 4092/4885TRPV6 1036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.