SCHEMBL3698799

SCHEMBL3698799

CNC(=O)OCc1cc(Sc2ccnc(OC)c2)n(-c2ccccc2Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 9/20 0.40
SLC16A1 P53985 8/20 0.40
ALDH1A1 P00352 1/20 0.37
CTSA P10619 1/20 0.35
PDE4B Q07343 1/20 0.34
SCN9A Q15858 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
BRAF P15056 1/20 0.33
NR3C2 P08235 1/20 0.33
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132130 0.83 SLC16A3 (0.38) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3709000 0.83 SLC16A3 (0.37) SLC16A3SLC16A1PDE4BNPC1HPGD
SCHEMBL3707729 0.83 SLC16A3 (0.46) SLC16A3SLC16A1PDE4BNPC1HPGD
SCHEMBL4132125 0.81 SLC16A3 (0.40) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3695878 0.79 PDE4B (0.46) ALDH1A1PDE4BNPC1HPGDRAB9A
SCHEMBL3700573 0.79 SLC16A3 (0.39) SLC16A3SLC16A1ALDH1A1CTSABRAF
SCHEMBL3700575 0.79 SLC16A3 (0.40) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3700571 0.78 HTR2C (0.47) SLC16A3SLC16A1ALDH1A1BRAF
SCHEMBL4126088 0.77 ALDH1A1 (0.35) SLC16A3SLC16A1ALDH1A1CTSAPDE4B
SCHEMBL3707175 0.73 SLC6A9 (0.33) TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed