SCHEMBL3701211

SCHEMBL3701211

C[C@@H]1CN(c2c(F)cc(C(=O)CF)cc2CO)C[C@H](C)O1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TSHR P16473 1/20 0.36
USP30 Q70CQ3 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HPGD P15428 1/20 0.34
NPC1 O15118 4/20 0.32
RAB9A P51151 3/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 2/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
MAPT P10636 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011006 0.78 KDM4E (0.39) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL3069796 0.72 KDM4E (0.38) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL2309750 0.72 TSHR (0.38) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL5014295 0.72 TSHR (0.37) ALDH1A1NPSR1TSHRUSP30KDM4E
SCHEMBL3066491 0.70 KDM4E (0.36) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL2307645 0.70 TSHR (0.36) ALDH1A1NPSR1TSHRUSP30KDM4E
SCHEMBL2305888 0.70 ALDH1A1 (0.45) ALDH1A1NPSR1KDM4EHSD17B10HPGD
SCHEMBL3751398 0.70 KDM4E (0.40) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL2306361 0.70 KDM4E (0.40) ALDH1A1NPSR1TSHRKDM4EHTT
SCHEMBL2357083 0.70 KDM4E (0.40) ALDH1A1NPSR1TSHRKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193132-A2 3-SPIROPYRIMIDINETRIONE-QUINOLINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AstraZeneca AB (SE) 2010-06-09 EP disclosed
WO-2009004382-A2 3-SPIROPYRIMIDINETRIONE-QUINOLINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2009-01-08 WO disclosed