SCHEMBL3701348

SCHEMBL3701348

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)C(F)C=O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.46
CASP7 P55210 2/20 0.46
CASP1 P29466 2/20 0.46
CASP9 P55211 2/20 0.46
MMP3 P08254 1/20 0.45
PSMB1 P20618 1/20 0.45
PSMB5 P28074 1/20 0.45
PSMB2 P49721 1/20 0.45
CTSL P07711 5/20 0.45
CTSK P43235 3/20 0.44
CAPN1 P07384 2/20 0.44
CTSB P07858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL157170 0.92 CAPN1 (0.47) CASP3CASP7CASP1CASP9MMP3
SCHEMBL31248471 0.90 CAPN1 (0.51) CASP3CASP7CASP1CASP9MMP3
SCHEMBL19190188 0.88 MMP3 (0.49) CASP3CASP7CASP1CASP9MMP3
SCHEMBL2034855 0.87 CAPN1 (0.48) CASP3CASP7CASP1CASP9MMP3
SCHEMBL3491057 0.83 PTPN1 (0.47) CASP3CASP7CASP1CASP9PSMB1
SCHEMBL9961858 0.82 CASP3 (0.65) CASP3CASP7CASP1CASP9CTSL
SCHEMBL7938093 0.80 CAPN1 (0.60) CTSLCTSKCAPN1CTSB
SCHEMBL20257154 0.80 REN (0.46) PSMB1PSMB5PSMB2CTSLCTSK
SCHEMBL23133281 0.80 REN (0.48) CTSLCTSKCAPN1CTSB
SCHEMBL20257155 0.80 REN (0.48) CTSLCTSKCAPN1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7838645-B2 comprising antibodies that specifically bind caspase-8 as inhibitors; cancer; activation of the receptor-interacting protein (RIP, a serine-threonine kinase) and Jun N-terminal kinase induce cell death with the morphology of autophagy UNIVERSITY OF MARYLAND COLLEGE PARK (US) 2010-11-23 US disclosed
US-20050276809-A1 comprising antibodies that specifically bind caspase-8 as inhibitors; cancer; activation of the receptor-interacting protein (RIP, a serine-threonine kinase) and Jun N-terminal kinase induce cell death with the morphology of autophagy NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-12-15 US disclosed