SCHEMBL3701586

SCHEMBL3701586

CCN(CC)C1CCN(c2nc(NCc3ccccc3)nc3nnc(-c4ccc(F)cc4)nc23)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 5/20 0.39
TLR7 Q9NYK1 4/20 0.39
PDE4A P27815 4/20 0.39
PDE4B Q07343 4/20 0.39
PDE4C Q08493 4/20 0.39
PDE4D Q08499 4/20 0.39
CCNE2 O96020 2/20 0.38
CCNA2 P20248 2/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
CCNA1 P78396 2/20 0.38
MAPK14 Q16539 1/20 0.37
HRH1 P35367 2/20 0.37
HRH4 Q9H3N8 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 1/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3786948 0.87 PDE4A (0.43) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3783454 0.85 ACHE (0.47) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3704626 0.85 HRH4 (0.52) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3704323 0.84 CCNE2 (0.40) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3781421 0.83 PDE4A (0.41) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3785003 0.83 PDE4A (0.47) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3779641 0.83 HTT (0.50) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL3788927 0.82 ACHE (0.44) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3784136 0.82 PDE4A (0.44) TLR9TLR7PDE4APDE4BPDE4C
SCHEMBL3781745 0.81 ACHE (0.38) TLR9TLR7PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed