SCHEMBL370200

SCHEMBL370200

COC(=O)c1cccc(C(CC(=O)c2ccc(=O)n(C)c2)c2ccc(Cl)cc2C)c1Oc1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.37
SCN8A Q9UQD0 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HPGD P15428 1/20 0.34
CTSA P10619 3/20 0.33
LMNA P02545 2/20 0.33
POLB P06746 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
F11 P03951 1/20 0.33
MAPK8 P45983 1/20 0.33
PTGER4 P35408 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370199 0.90 BRD4 (0.39) BRD4CYP1A2CYP2C19ALDH1A1MEN1
SCHEMBL370635 0.88 BRD4 (0.40) BRD4MEN1KMT2AMAPTTDP1
SCHEMBL370383 0.85 CYP1A2 (0.36) CYP1A2CYP2C19ALDH1A1MEN1KMT2A
SCHEMBL368800 0.83 FFAR1 (0.35) CYP1A2CYP2C19ALDH1A1KMT2AHPGD
SCHEMBL370636 0.80 BRD4 (0.37) BRD4LMNAPTGER4
SCHEMBL369275 0.80 P2RX3 (0.39) CYP1A2CYP2C19ALDH1A1LMNAPOLB
SCHEMBL1390419 0.78 LMNA (0.43) CYP1A2CYP2C19MEN1KMT2ALMNA
SCHEMBL1390299 0.78 TDP1 (0.33) BRD4ALDH1A1KMT2AHPGDCTSA
SCHEMBL1390202 0.77 KMT2A (0.35) BRD4ALDH1A1MEN1KMT2ACTSA
SCHEMBL368801 0.76 P2RX3 (0.42) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed