SCHEMBL370383

SCHEMBL370383

COC(=O)c1ccc(C(CC(=O)c2ccc(=O)n(C)c2)c2ccc(Cl)cc2C)c(Oc2ccccc2)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KDM4E B2RXH2 2/20 0.34
LMNA P02545 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
NPBWR1 P48145 1/20 0.32
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
F11 P03951 2/20 0.31
CREBBP Q92793 1/20 0.31
GAA P10253 1/20 0.31
F10 P00742 1/20 0.31
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370200 0.85 BRD4 (0.37) CYP1A2CYP2C19ALDH1A1KMT2AMEN1
SCHEMBL368800 0.82 FFAR1 (0.35) CYP1A2CYP2C19ALDH1A1KMT2AHPGD
SCHEMBL369275 0.82 P2RX3 (0.39) CYP1A2CYP2C19ALDH1A1KDM4ELMNA
SCHEMBL370199 0.81 BRD4 (0.39) CYP1A2CYP2C19ALDH1A1KMT2AMEN1
SCHEMBL368801 0.79 P2RX3 (0.42) LMNAL3MBTL1CREBBP
SCHEMBL1390419 0.79 LMNA (0.43) CYP1A2CYP2C19KMT2AMEN1LMNA
SCHEMBL370635 0.78 BRD4 (0.40) KMT2AMEN1TDP1
SCHEMBL1390202 0.78 KMT2A (0.35) ALDH1A1KMT2AMEN1TDP1
SCHEMBL370636 0.77 BRD4 (0.37) LMNAL3MBTL1
SCHEMBL369771 0.76 P2RX3 (0.37) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed