SCHEMBL3702296

SCHEMBL3702296

COc1cccc(C(=O)N[C@H]2CC[C@H](N3CCN(C)CC3)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
TSHR P16473 2/20 0.61
MCHR1 Q99705 4/20 0.55
NPC1 O15118 2/20 0.54
GRM5 P41594 1/20 0.54
LMNA P02545 4/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MAPT P10636 1/20 0.53
HTT P42858 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MAPK1 P28482 1/20 0.53
CCR3 P51677 1/20 0.52
KDM4E B2RXH2 1/20 0.52
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51
CHRM1 P11229 1/20 0.51
USP2 O75604 1/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29363800 0.88 ALDH1A1 (0.72) ALDH1A1TSHRMCHR1NPC1GRM5
SCHEMBL4516387 0.88 ALDH1A1 (0.72) ALDH1A1TSHRMCHR1NPC1GRM5
SCHEMBL17706078 0.88 ALDH1A1 (0.58) ALDH1A1TSHRMCHR1NPC1GRM5
SCHEMBL2468483 0.85 NPC1 (0.71) ALDH1A1TSHRMCHR1NPC1GRM5
SCHEMBL17706081 0.84 MCHR1 (0.68) ALDH1A1MCHR1LMNASMN1; SMN2MAPT
SCHEMBL14246914 0.83 DRD2 (0.64) ALDH1A1TSHRGRM5LMNASMN1; SMN2
SCHEMBL14246915 0.83 DRD2 (0.64) ALDH1A1TSHRGRM5LMNASMN1; SMN2
SCHEMBL1667825 0.80 RAB9A (0.73) ALDH1A1TSHRNPC1GRM5LMNA
SCHEMBL17993402 0.80 ALDH1A1 (0.66) ALDH1A1TSHRLMNAKDM4E
SCHEMBL12893788 0.80 HTR4 (0.48) ALDH1A1MCHR1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205603-A1 PYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS Cyclacel Limited (GB) 2010-07-14 EP disclosed
WO-2009040556-A1 PYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS CYCLACEL LIMITED (GB) 2009-04-02 WO disclosed