SCHEMBL3703498

SCHEMBL3703498

CCOc1ccc(C2CCCc3cc(OC)ccc3C2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP24A1 Q07973 6/20 0.48
CYP27A1 Q02318 3/20 0.48
CYP26A1 O43174 3/20 0.46
CYP19A1 P11511 2/20 0.46
METAP1 P53582 3/20 0.43
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
MPO P05164 1/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
MAPK1 P28482 1/20 0.41
KCNH2 Q12809 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13885522 0.90 CYP24A1 (0.48) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL3654990 0.90 CYP24A1 (0.48) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL9995721 0.85 CYP24A1 (0.47) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL5077391 0.85 CYP19A1 (0.57) CYP24A1CYP27A1CYP26A1CYP19A1DRD2
SCHEMBL16567983 0.85 MAOA (0.48) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL15012851 0.83 PTGS2 (0.44) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL6669546 0.82 CYP24A1 (0.53) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL15012600 0.81 GID4 (0.61) CYP24A1CYP27A1CYP26A1CYP19A1DRD2
SCHEMBL9995684 0.81 SLC6A2 (0.49) CYP24A1CYP27A1CYP26A1CYP19A1METAP1
SCHEMBL9995652 0.81 CYP24A1 (0.47) CYP24A1CYP27A1CYP26A1CYP19A1METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200962-A1 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY Bayer Schering Pharma Aktiengesellschaft (DE) 2010-06-30 EP claimed
WO-2009047343-A1 BENZOCYCLOHEPTENE DERIVATIVES AS ESTROGENS HAVING SELECTIVE ACTIVITY BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-04-16 WO claimed