SCHEMBL3705969

SCHEMBL3705969

COc1cccc(S(=O)(=O)c2cc(CN(CC(C)(C)C)C(=O)O)nn2-c2cccnc2F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 10/20 0.39
SLC16A1 P53985 8/20 0.39
NFE2L2 Q16236 4/20 0.37
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
MET P08581 1/20 0.34
MCTS1 Q9ULC4 1/20 0.34
CHRM5 P08912 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
MMP13 P45452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3700744 0.90 PTGDR2 (0.33) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL476415 0.89 HTR6 (0.35) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL3697999 0.89 P2RX7 (0.33) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL476339 0.89 HTR6 (0.32)
SCHEMBL4125764 0.88 NFE2L2 (0.40) SLC16A3SLC16A1NFE2L2METTAS2R14
SCHEMBL476326 0.87 COMT (0.36) PTGDR2
SCHEMBL476395 0.86 NAMPT (0.33)
SCHEMBL3697762 0.84 KDM4E (0.33) SLC16A3SLC16A1ABCC9ABCC8KCNJ11
SCHEMBL3705968 0.84 SLC16A3 (0.39) SLC16A3SLC16A1NFE2L2ABCC9ABCC8
SCHEMBL3703141 0.84 CA1 (0.44) SLC16A3SLC16A1NFE2L2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed