SCHEMBL3708683

SCHEMBL3708683

NC1(Cc2cccc(Cl)c2)CCC(=O)NC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
AKT2 P31751 1/20 0.42
MAOB P27338 3/20 0.40
MAOA P21397 2/20 0.40
PNMT P11086 2/20 0.40
KMT2A Q03164 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
MDM2 Q00987 1/20 0.38
CYP3A4 P08684 2/20 0.37
IDO1 P14902 2/20 0.37
AGXT P21549 2/20 0.37
HSD11B1 P28845 1/20 0.37
DAO P14920 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2473095 0.78 MAOA (0.59) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL3708719 0.78 MAPT (0.39) MAPTCYP2C9CYP2C19MAOBMAOA
Hydrochloric Acid SCHEMBL21879608 0.77 MAOB (0.57) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL5218251 0.76 PNMT (0.50) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL9667972 0.76 SLC6A4 (0.50) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL12585406 0.75 AKT2 (0.49) MAPTCYP2C9CYP2C19AKT2MAOB
Formic Acid SCHEMBL6207884 0.74 MAOA (0.49) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL6430626 0.71 AKT2 (0.46) MAPTAKT2MAOBMAOAPNMT
SCHEMBL208131 0.67 AOC3 (0.43) AKT2MAOBMAOAPNMTTAAR1
SCHEMBL2470610 0.66 SSTR1 (0.49) PNMTKMT2ATAAR1CYP3A4IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391603-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086251-A1 AROYLAMINO - AND HETEROAROYLAMINO-SUBSTITUTED PIPERIDINES AS GLYT-1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed