SCHEMBL3708765

SCHEMBL3708765

CCCCNc1cccc(-c2cccc(C(N)=O)c2)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
PARP1 P09874 3/20 0.40
BAZ2B Q9UIF8 1/20 0.40
BAZ2A Q9UIF9 1/20 0.40
DYRK1A Q13627 1/20 0.39
PRKCI P41743 1/20 0.39
FYN P06241 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
F3 P13726 1/20 0.39
CSF1R P07333 1/20 0.39
FLT1 P17948 1/20 0.39
FLT3 P36888 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SHMT1 P34896 1/20 0.38
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3704899 0.93 PARP1 (0.42) FAAHPARP1BAZ2BBAZ2ADYRK1A
SCHEMBL3698515 0.87 PARP1 (0.44) PARP1BAZ2BBAZ2ADYRK1APRKCI
SCHEMBL3714031 0.81 AR (0.48) BAZ2BBAZ2AFYNKDM4EALDH1A1
SCHEMBL6432991 0.78 NR1H4 (0.45) AKR1C3AKR1C2
SCHEMBL5647187 0.74 CNR2 (0.40) SMN1; SMN2ALDH1A1HPGD
SCHEMBL19710767 0.74 HTR7 (0.55) SMN1; SMN2PARP1F3HPGD
SCHEMBL3135455 0.74 PARP1 (0.53) PARP1BAZ2BBAZ2ADYRK1APRKCI
Hydrochloric Acid SCHEMBL29287792 0.73 PARP1 (0.51) PARP1BAZ2BBAZ2ADYRK1APRKCI
Hydrochloric Acid SCHEMBL29287827 0.73 PARP1 (0.51) PARP1BAZ2BBAZ2ADYRK1APRKCI
SCHEMBL3701695 0.73 PARP1 (0.51) PARP1BAZ2BBAZ2ADYRK1APRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed