SCHEMBL3714031

SCHEMBL3714031

Cc1c(NCc2ccccc2)cccc1-c1cccc(C(N)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.48
CD38 P28907 1/20 0.46
PLA2G2A P14555 1/20 0.46
RET P07949 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HDAC8 Q9BY41 3/20 0.45
SHMT1 P34896 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
CDC7 O00311 1/20 0.44
ROCK2 O75116 1/20 0.44
MAP4K4 O95819 1/20 0.44
GSK3B P49841 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CFD P00746 1/20 0.43
FYN P06241 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698515 0.85 PARP1 (0.44) RETSHMT1MKNK2BAZ2BBAZ2A
SCHEMBL3704899 0.82 PARP1 (0.42) RETHDAC8SHMT1BAZ2BBAZ2A
SCHEMBL3708765 0.81 FAAH (0.43) KDM4EALDH1A1HPGDSHMT1FYN
SCHEMBL16438662 0.76 ALDH1A1 (0.49) ALDH1A1HPGDCDC7ROCK2GSK3B
SCHEMBL6432991 0.75 NR1H4 (0.45) PLA2G2AROCK2
SCHEMBL3714028 0.74 ALDH1A1 (0.46) ARCD38KDM4EALDH1A1HPGD
SCHEMBL3135455 0.74 PARP1 (0.53) FYNBAZ2BBAZ2A
SCHEMBL5307077 0.73 PARP1 (0.56) PLA2G2ACDC7ROCK2GSK3BCLK4
SCHEMBL12497396 0.73 APP (0.65) ALDH1A1CDC7ROCK2MAP4K4GSK3B
Hydrochloric Acid SCHEMBL29287827 0.73 PARP1 (0.51) BAZ2BBAZ2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed