SCHEMBL3698515

SCHEMBL3698515

CCNc1cccc(-c2cccc(C(N)=O)c2)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.44
BAZ2B Q9UIF8 1/20 0.43
BAZ2A Q9UIF9 1/20 0.43
PGK1 P00558 1/20 0.43
PRKCI P41743 1/20 0.42
DYRK1A Q13627 1/20 0.42
CSF1R P07333 1/20 0.41
FLT1 P17948 1/20 0.41
FLT3 P36888 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
RORC P51449 1/20 0.41
ERN1 O75460 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
SHMT1 P34896 1/20 0.40
BRD4 O60885 2/20 0.40
CREBBP Q92793 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3704899 0.90 PARP1 (0.42) PARP1BAZ2BBAZ2APRKCIDYRK1A
SCHEMBL3708765 0.87 FAAH (0.43) PARP1BAZ2BBAZ2APRKCIDYRK1A
SCHEMBL3714031 0.85 AR (0.48) BAZ2BBAZ2AMKNK2SHMT1RET
SCHEMBL27789898 0.83 KDR (0.49)
SCHEMBL3135455 0.78 PARP1 (0.53) PARP1BAZ2BBAZ2APRKCIDYRK1A
Hydrochloric Acid SCHEMBL29287792 0.77 PARP1 (0.51) PARP1BAZ2BBAZ2APRKCIDYRK1A
SCHEMBL3701695 0.77 PARP1 (0.51) PARP1BAZ2BBAZ2APRKCIDYRK1A
Hydrochloric Acid SCHEMBL29287827 0.77 PARP1 (0.51) PARP1BAZ2BBAZ2APRKCIDYRK1A
SCHEMBL6432991 0.76 NR1H4 (0.45) AKR1C3AKR1C2
SCHEMBL16438662 0.74 ALDH1A1 (0.49) PARP1BAZ2BBAZ2APRKCIDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed