SCHEMBL3711244

SCHEMBL3711244

CCOC(=O)c1cc(-c2ccco2)nc(-c2ccc(C#Cc3cccnc3)cc2)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.45
KDM4E B2RXH2 9/20 0.45
HPGD P15428 6/20 0.45
GAA P10253 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 8/20 0.44
USP2 O75604 4/20 0.44
MAPT P10636 7/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
HSD17B10 Q99714 3/20 0.43
TSHR P16473 2/20 0.43
GLA P06280 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
MCL1 Q07820 11/20 0.43
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3716537 0.91 MCL1 (0.47) ALDH1A1KDM4EHPGDGAAPOLB
SCHEMBL3713520 0.89 GRM5 (0.46) ALDH1A1KDM4EHPGDGAASMN1; SMN2
SCHEMBL13188547 0.86 MCL1 (0.47) ALDH1A1KDM4EMEN1KMT2AMCL1
SCHEMBL3712449 0.86 GRM5 (0.44) ALDH1A1KDM4EHPGDGAASMN1; SMN2
SCHEMBL3713434 0.86 GRM5 (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTMEN1
SCHEMBL3713522 0.85 GRM5 (0.43) ALDH1A1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL3710606 0.83 GRM5 (0.42) ALDH1A1KDM4EHPGDSMN1; SMN2POLB
SCHEMBL3720526 0.83 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDGAASMN1; SMN2
SCHEMBL3710598 0.80 GRM5 (0.42) ALDH1A1KDM4EHPGDSMN1; SMN2MAPT
SCHEMBL3709730 0.77 PLA2G2A (0.44) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed